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Introduction:
Tramadol, a versatile opioid analgesic, has carved a niche in the realm of pain management. Distinctive in its pharmacological profile, Tramadol combines opioid receptor binding with the inhibition of serotonin and norepinephrine reuptake.
Pharmacology: The Dual Dance of Opioid and Non-Opioid Pathways:
Opioid Receptor Binding: Tramadol's primary mechanism involves binding to mu-opioid receptors in the central nervous system, dampening the transmission of pain signals and modulating the perception of pain.
Serotonin and Norepinephrine Reuptake Inhibition: Beyond its opioid action, Tramadol inhibits the reuptake of serotonin and norepinephrine, contributing to its unique analgesic effects and potential benefits in neuropathic pain.
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